Yous, Said: search on Z-Library

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1

Pictet–Spengler heterocyclizations via microwave-assisted degradation of DMSO

Christophe Mésangeau, Saïd Yous, Basile Pérès, Daniel Lesieur, Thierry Besson

Journal:

Tetrahedron Letters

Year:

2005

Language:

english

File:

PDF, 114 KB

english, 2005

2

Design and synthesis of 2,6-disubstituted-8-amino imidazo[1,2a]pyridines, a promising privileged structure

Boulahjar, Rajaa, Arias, Angela Rincon, Bolteau, Raphaël, Renault, Nicolas, Coevoet, Mathilde, Barczyk, Amélie, Duroux, Romain, Yous, Saïd, Melnyk, Patricia, Agouridas, Laurence

Journal:

Bioorganic & Medicinal Chemistry

Year:

2018

Language:

english

File:

PDF, 1013 KB

english, 2018

3

Quantitative structure-activity relationships studies of antioxidant hexahydropyridoindoles and flavonoid derivatives

Durand, Anne-Catherine, Farce, Amaury, Carato, Pascal, Dilly, Sebastien, Yous, Said, Berthelot, Pascal, Chavatte, Philippe

Journal:

Journal of Enzyme Inhibition and Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 133 KB

english, 2007

4

Synthesis of 6-(2,2-Dimethyl-3,4-dihydro-3-oxo-1,4 (2H)-benzoxazin-7-yl)pyridazin-3-ones.

Ziaeddin Moussavi, Nicolas Lebegue, Pascal Carato, Said Yous, Pascal Berthelot

Journal:

Year:

2004

File:

PDF, 24 KB

2004

5

A new synthesis of N-alkyl pyrazolidine-3,5-diones and tetrahydropyridazine-3,6-diones

Bertrand Le Bourdonnec, Emmanuelle Meulon, Saïd Yous, Raymond Houssin, Jean-Pierre Hénichart

Journal:

Journal of Heterocyclic Chemistry

Year:

2000

File:

PDF, 335 KB

2000

6

Novel 2(3H)-Benzothiazolones as Highly Potent and Selective Sigma-1 Receptor Ligands

Saïd Yous, Valérie Wallez, Mirabelle Belloir, Daniel H. Caignard, Christopher R. McCurdy, Jacques H. Poupaert

Journal:

Medicinal Chemistry Research

Year:

2005

File:

PDF, 335 KB

2005

7

Synthesis and Pharmacological Evaluation of New Pyrazolidine-3,5-diones as AT 1 Angiotensin II Receptor Antagonists

Le Bourdonnec, Bertrand, Meulon, Emmanuelle, Yous, Saïd, Goossens, Jean-François, Houssin, Raymond, Hénichart, Jean-Pierre

Journal:

Journal of Medicinal Chemistry

Year:

2000

Language:

english

File:

PDF, 179 KB

english, 2000

8

Lipid-lowering properties of 6-benzoyl-2(3 H )-benzothiazolone and structurally related compounds

Yous, SaÏd, Lebegue, Nicolas, Poupaert, Jacques-henry, Chavatte, Philippe, Berthelot, Pascal

Journal:

Journal of Enzyme Inhibition and Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 300 KB

english, 2005

9

A mild and efficient route to 2-benzyl tryptamine derivatives via ring-opening of β-carbolines

Fariza Hadjaz, Saïd Yous, Nicolas Lebegue, Pascal Berthelot, Pascal Carato

Journal:

Year:

2008

Language:

english

File:

PDF, 204 KB

english, 2008

10

Antioxydant activity of β-carboline derivatives in the LDL oxidation model

Fariza Hadjaz, Soizic Besret, Françoise Martin-Nizard, Saïd Yous, Sébastien Dilly, Nicolas Lebegue, Philippe Chavatte, Patrick Duriez, Pascal Berthelot, Pascal Carato

Journal:

European Journal of Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 614 KB

english, 2011

11

Homology modelling of the serotoninergic 5-HT 2c receptor

Farce, Amaury, Dilly, Sebastien, Yous, Said, Berthelot, Pascal, Chavatte, Philippe

Journal:

Journal of Enzyme Inhibition and Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 1024 KB

english, 2006

12

Design of experiments for enantiomeric separation in supercritical fluid chromatography

Landagaray, Elodie, Vaccher, Claude, Yous, Saïd, Lipka, Emmanuelle

Journal:

Journal of Pharmaceutical and Biomedical Analysis

Year:

2015

Language:

english

File:

PDF, 943 KB

english, 2015

13

Friedel-Crafts Acylation of 2(3H)-Benzoxazolone: Investigation of the Role of the Catalyst and Microwave Activation

Messaoud Liacha, Saïd Yous, Jacques H. Poupaert, Patrick Depreux, Hocine Aichaoui

Journal:

Monatshefte für Chemie - Chemical Monthly

Year:

1999

Language:

english

File:

PDF, 72 KB

english, 1999

14

ChemInform Abstract: Absolute Configuration of N-[(-)-2-(7-Methoxy-1,2,3,4-tetrahydro-1-naphthyl)ethyl] cyclopropylcarboxamide, a Highly Potent and Selective Melatonin Analogue.

Abdelhalim Guelzim, Emmanuelle Belloli, Said Yous, Claude Vaccher

Journal:

Year:

2001

File:

PDF, 29 KB

2001

15

Synthesis of 2-(Ethylsulfanyl)aniline Derivatives Through the Unexpected Ring Opening of N-Substituted-2(3H)-benzothiazolones.

Nicolas Lebegue, Gaetan Charrier, Pascal Carato, Said Yous, Pascal Berthelot

Journal:

Year:

2005

File:

PDF, 20 KB

2005

16

Efficient and selective deprotection method for N-protected 2(3H)-benzoxazolones and 2(3H)-benzothiazolones

Pascal Carato, Saïd Yous, Didier Sellier, Jacques H. Poupaert, Nicolas Lebegue, Pascal Berthelot

Journal:

Year:

2004

Language:

english

File:

PDF, 119 KB

english, 2004

17

Quantification of the water/lipid affinity of melatonin and a pinoline derivative in lipid models

Jamila Mekhloufi, Heidi Vitrac, Saïd Yous, Patrick Duriez, Daniel Jore, Monique Gardès-Albert, Dominique Bonnefont-Rousselot

Journal:

Journal of Pineal Research

Year:

2007

Language:

english

File:

PDF, 595 KB

english, 2007

18

Synthesis and Evaluation of Benzoxazolinonic Imidazoles and Derivatives as Non-steroidal Aromatase Inhibitors

Nativelle-Serpentini, Celine, Moslemi, Safa, Yous, Said, Ha Park, Chang, Lesieur, Daniel, Sourdaine, Pascal, Séralini, Gilles-Eric

Journal:

Journal of Enzyme Inhibition and Medicinal Chemistry

Year:

2004

Language:

english

File:

PDF, 207 KB

english, 2004

19

Design and synthesis of fused tetrahydroisoquinoline-iminoimidazolines

Moas-Héloire, Valeria, Renault, Nicolas, Batalha, Vania, Arias, Angela Rincon, Marchivie, Mathieu, Yous, Said, Deguine, Noémie, Buée, Luc, Chavatte, Philippe, Blum, David, Lopes, Luisa, Melnyk, Patric

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 1.38 MB

english, 2015

20

Three-Dimensional Quantitative Structure-Activity Relationship of Arylalkylamine N-acetyltransferase (AANAT) Inhibitors: A Comparative Molecular Field Analysis

Philippe Chavatte, Saïd Yous, Nathalie Beaurain, Christophe Mésangeau, Gilles Ferry, Daniel Lesieur

Journal:

Molecular Informatics

Year:

2001

Language:

english

File:

PDF, 181 KB

english, 2001

21

Antioxidant activity of benzoxazolinonic and benzothiazolinonic derivatives in the LDL oxidation model

Ismaël Yekini, Fatma Hammoudi, Françoise Martin-Nizard, Saïd Yous, Nicolas Lebegue, Pascal Berthelot, Pascal Carato

Journal:

Bioorganic & Medicinal Chemistry

Year:

2009

Language:

english

File:

PDF, 288 KB

english, 2009

22

Characterization of the melatoninergic MT3 binding site on the NRH:quinone oxidoreductase 2 enzyme

François Mailliet, Gilles Ferry, Fanny Vella, Sylvie Berger, Francis Cogé, Pascale Chomarat, Catherine Mallet, Sophie-Pénélope Guénin, Gérald Guillaumet, Marie-Claude Viaud-Massuard, Saïd Yous, Philip

Journal:

Biochemical Pharmacology

Year:

2005

Language:

english

File:

PDF, 546 KB

english, 2005

23

Design and Synthesis of Naphthalenic Dimers as Selective MT1 Melatoninergic Ligands

Descamps-François, Carole, Yous, Saïd, Chavatte, Philippe, Audinot, Valérie, Bonnaud, Anne, Boutin, Jean A., Delagrange, Philippe, Bennejean, Caroline, Renard, Pierre, Lesieur, Daniel

Journal:

Journal of Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 47 KB

english, 2003

24

New phenylaniline derivatives as modulators of amyloid protein precursor metabolism

Gay, Marion, Carato, Pascal, Coevoet, Mathilde, Renault, Nicolas, Larchanché, Paul-Emmanuel, Barczyk, Amélie, Yous, Saïd, Buée, Luc, Sergeant, Nicolas, Melnyk, Patricia

Journal:

Bioorganic & Medicinal Chemistry

Year:

2018

Language:

english

File:

PDF, 1.58 MB

english, 2018

25

Synthesis of 2(3H)-Benzoxazolone Derivatives as Potential Melatonin Receptor Ligands.

Christophe Mesangeau, Jacques H. Poupaert, Pascal Carato, Said Yous

Journal:

Year:

2004

File:

PDF, 78 KB

2004

26

Synthesis and pharmacological evaluation of dual ligands for melatonin (MT1/MT2) and serotonin 5-HT2C receptor subtypes (II)

Ettaoussi, Mohamed, Pérès, Basile, Errazani, Aïcha, Boutin, Jean A., Caignard, Daniel-Henri, Delagrange, Philippe, Melnyk, Patricia, Berthelot, Pascal, Yous, Saïd

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 653 KB

english, 2015

27

Synthesis of 2(3H)-Benzoxazolone Derivatives as Potential Melatonin Receptor Ligands

Carato, Pascal, Mésangeau, Christophe, H. Poupaert, Jacques, Yous, Saïd

Journal:

Year:

2003

Language:

english

File:

PDF, 66 KB

english, 2003

28

On the reaction of meldrum's acid with N-trimethylsilylanilines substituted by electron withdrawing groups

Sandrine Roche, Saïd Yous, Daniel Couturier, Benoît Rigo

Journal:

Journal of Heterocyclic Chemistry

Year:

1999

File:

PDF, 180 KB

1999

29

Preparation and pharmacological evaluation of a novel series of 2-(phenylthio)benzo[b]thiophenes as selective MT2 receptor ligands

Christophe Mésangeau, Mikaël Fraise, Philippe Delagrange, Daniel Henri Caignard, Jean Albert Boutin, Pascal Berthelot, Saïd Yous

Journal:

European Journal of Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 243 KB

english, 2011

30

Synthesis of 6- and 7-acyl-4H-benzothiazin-3-ones

Pascal Carato, Ziaeddine Moussavi, Ahmed Sabaouni, Nicolas Lebegue, Pascal Berthelot, Saïd Yous

Journal:

Year:

2006

Language:

english

File:

PDF, 172 KB

english, 2006

31

Synthesis of Nitroindole Derivatives with High Affinity and Selectivity for Melatoninergic Binding Sites MT 3

Leclerc, Véronique, Yous, Saïd, Delagrange, Philippe, Boutin, Jean A., Renard, Pierre, Lesieur, Daniel

Journal:

Journal of Medicinal Chemistry

Year:

2002

Language:

english

File:

PDF, 82 KB

english, 2002

32

New Access to 5-Substituted 1,3-Benzothiazol-2(3H)-ones and Their N-Methyl Analogues by a Palladium Coupling Reaction

Pirat, Céline, Ultré, Vincent, Lebegue, Nicolas, Berthelot, Pascal, Yous, Saïd, Carato, Pascal

Journal:

Year:

2011

Language:

english

File:

PDF, 102 KB

english, 2011

33

Interactions of bexarotene (LGD1069, Targretin) with the coagulation system

Anne Hespel, Najet Mejdoubi-Charef, Said Yous, José Courty, Dulce Papy-Garcia, Said Charef

Journal:

Cancer Chemotherapy and Pharmacology

Year:

2011

Language:

english

File:

PDF, 1.65 MB

english, 2011

34

Efficient and Selective Deprotection Method for N-Protected 2(3H)-Benzoxazolones and 2(3H)-Benzothiazolones.

Pascal Carato, Said Yous, Didier Sellier, Jacques H. Poupaert, Nicolas Lebegue, Pascal Berthelot

Journal:

Year:

2005

File:

PDF, 23 KB

2005

35

Synthesis of 2-(ethylsulfanyl)aniline derivatives through the unexpected ring opening of N-substituted-2(3H)-benzothiazolones

Nicolas Lebegue, Gaetan Charrier, Pascal Carato, Saïd Yous, Pascal Berthelot

Journal:

Tetrahedron Letters

Year:

2004

Language:

english

File:

PDF, 251 KB

english, 2004

36

Synthesis and biological evaluation of new naphtho- and quinolinocyclopentane derivatives as potent melatoninergic (MT 1 /MT 2 ) and serotoninergic (5-HT 2C ) dual ligands

Duroux, Romain, Rami, Marouan, Landagaray, Elodie, Ettaoussi, Mohamed, Caignard, Daniel-Henri, Delagrange, Philippe, Melnyk, Patricia, Yous, Saïd

Journal:

European Journal of Medicinal Chemistry

Year:

2017

Language:

english

File:

PDF, 739 KB

english, 2017

37

Design and synthesis of benzofuranic derivatives as new ligands at the melatonin-binding site MT3

Mohamed Ettaoussi, Basile Péres, Fréderique Klupsch, Philippe Delagrange, Jean-A. Boutin, Pierre Renard, Daniel-H. Caignard, Philippe Chavatte, Pascal Berthelot, Daniel Lesieur, Saïd Yous

Journal:

Bioorganic & Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 188 KB

english, 2008

38

Design and synthesis of naphthalenic derivatives as new ligands at the melatonin binding site MT3

Véronique Leclerc, Mohamed Ettaoussi, Marouan Rami, Amaury Farce, Jean Albert Boutin, Philippe Delagrange, Daniel-Henri Caignard, Pierre Renard, Pascal Berthelot, Saïd Yous

Journal:

European Journal of Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 309 KB

english, 2011

39

Old and new inhibitors of quinone reductase 2

Gilles Ferry, Sabrina Hecht, Sylvie Berger, Natacha Moulharat, Francis Coge, Gérald Guillaumet, Véronique Leclerc, Saïd Yous, Philippe Delagrange, Jean A. Boutin

Journal:

Chemico-Biological Interactions

Year:

2010

Language:

english

File:

PDF, 467 KB

english, 2010

40

Antagonists of the adenosine A 2A receptor based on a 2-arylbenzoxazole scaffold: Investigation of the C5- and C7-positions to enhance affinity

Duroux, Romain, Agouridas, Laurence, Renault, Nicolas, El Bakali, Jamal, Furman, Christophe, Melnyk, Patricia, Yous, Saïd

Journal:

European Journal of Medicinal Chemistry

Year:

2018

Language:

english

File:

PDF, 1.50 MB

english, 2018

41

Three-Dimensional Quantitative Structure−Activity Relationships of Cyclo-oxygenase-2 (COX-2) Inhibitors: A Comparative Molecular Field Analysis

Chavatte, Philippe, Yous, Saïd, Marot, Christophe, Baurin, Nicolas, Lesieur, Daniel

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 337 KB

english, 2001

42

Melatonergic ligands: Design, synthesis and pharmacological evaluation of novel series of naphthofuranic derivatives

Landagaray, Elodie, Ettaoussi, Mohamed, Duroux, Romain, Boutin, Jean A., Caignard, Daniel-Henri, Delagrange, Philippe, Melnyk, Patricia, Berthelot, Pascal, Yous, Saïd

Journal:

European Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 557 KB

english, 2016

43

Bitopic Fluorescent Antagonists of the A 2A Adenosine Receptor Based on Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine Functionalized Congeners

Duroux, Romain, Ciancetta, A., Mannes, Philip, Yu, Jinha, Boyapati, Shireesha, Gizewski, Elizabeth, Yous, Said, Ciruela, Francisco, Auchampach, John, Gao, Zhan-Guo, Jacobson, Kenneth

Journal:

Year:

2017

Language:

english

File:

PDF, 2.04 MB

english, 2017

44

ChemInform Abstract: Synthesis of 6-Chloromethyl Benzothiazolin-2-one and of 6-Chloromethyl Benzoxazolin-2-one.

Pascal Carato, Said Yous, Patrick Depreux

Journal:

Year:

2000

File:

PDF, 31 KB

2000

45

ChemInform Abstract: Friedel—Crafts Acylation of 2(3H)-Benzoxazolone: Investigation of the Role of the Catalyst and Microwave Activation.

Messaoud Liacha, Said Yous, Jacques H. Poupaert, Patrick Depreux, Hocine Aichaoui

Journal:

Year:

2000

File:

PDF, 30 KB

2000

46

Three-Dimensional Quantitative Structure–Activity Relationship of MT3 Melatonin Binding Site Ligands: A Comparative Molecular Field Analysis

Amaury Farce, Sébastien Dilly, Ahmed Sabaouni, Saïd Yous, Pascal Berthelot, Jean A. Boutin, Philippe Delagrange, Pierre Renard, Philippe Chavatte

Journal:

Molecular Informatics

Year:

2007

Language:

english

File:

PDF, 314 KB

english, 2007

47

SYNTHESIS OF 6-CHLOROMETHYL BENZOTHIAZOLIN-2-ONE AND OF 6-CHLOROMETHYL BENZOXAZOLIN-2-ONE

Carato, Pascal, Yous, Saïd, Depreux, Patrick

Journal:

Organic Preparations and Procedures International

Year:

2000

Language:

english

File:

PDF, 367 KB

english, 2000

48

New Radioligands for Describing the Molecular Pharmacology of MT1 and MT2 Melatonin Receptors

Legros, Céline, Matthey, Ulrich, Grelak, Teresa, Pedragona-Moreau, Sandrine, Hassler, Werner, Yous, Saïd, Thomas, Emmanuel, Suzenet, Franck, Folleas, Benoît, Lefoulon, François, Berthelot, Pascal, Cai

Journal:

International Journal of Molecular Sciences

Year:

2013

Language:

english

File:

PDF, 438 KB

english, 2013

49

Design, synthesis and evaluation of 2-aryl benzoxazoles as promising hit for the A 2A receptor

Duroux, Romain, Renault, Nicolas, Cuelho, Joana Esteves, Agouridas, Laurence, Blum, David, Lopes, Luisa V., Melnyk, Patricia, Yous, Saïd

Journal:

Journal of Enzyme Inhibition and Medicinal Chemistry

Year:

2017

Language:

english

File:

PDF, 1.96 MB

english, 2017

50

Carbazole scaffolds in cancer therapy: a review from 2012 to 2018

Issa, Samar, Prandina, Anthony, Bedel, Nicolas, Rongved, Pål, Yous, Saïd, Le Borgne, Marc, Bouaziz, Zouhair

Journal:

Journal of Enzyme Inhibition and Medicinal Chemistry

Year:

2019

Language:

english

File:

PDF, 6.53 MB

english, 2019

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